Stable isotope

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Macimorelin acetate

CAS #

945212-59-9

Packing size

5mg, 10mg, 100mg, bulk (gram scale)

Synonyme(s)

Macrilen, ARD-07, AEZS-130, JMV1843

Therapeutic Drug Monitoring (TDM)Analytical Standards

Macimorelin acetate (Macrilen) is a Growth Hormone Secretagogue (GHS) causing the release of Growth Hormone (GH) from the pituitary gland. It became the first EMEA (2019) and FDA (2017) approved GHS to diagnose Adult GH Deficiency (AGHD). Macimorelin boasts an oral formulation for ease of administration for patients and providers. Macimorelin is a mimic of ghrelin, a growth hormone secretagogue (GHS or GHRP). It binds to the growth hormone secretagogue receptor (GHSR) causing release of growth hormone from the pituitary gland.

Aspect

White solid

Purity

98%

Solubility

methanol, water, acetonitrile

Molecular weight

534,62

Molecular formula

C₂₈H₃₄N₆O₅

IUPAC

1-(((R)-1-(((R)-1-formamido-2-(1H-indol-3-yl)ethyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)amino)-2-methyl-1-oxopropan-2-aminium acetate

J. M. Garcia et al., J. Clin. Endocrinol. Metab., 2018, 103, 8, 3083-3093. read article

Macimorelin acetate

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